In Vitro ADME Services

Comprehensive in vitro ADME studies that help teams evaluate metabolism, permeability, distribution, and drug interaction potential early in the drug discovery process.

From physicochemical characterization and metabolic stability testing to transporter studies and metabolite identification, BioDuro generates the data needed to identify potential liabilities, optimize compounds, and support confident candidate selection across small molecules, peptides, PROTACs, ADCs, and oligonucleotide therapeutics.

In Vitro ADME Support for Discovery Programs

BioDuro provides in vitro ADME services designed to help researchers better understand compound disposition, identify potential liabilities earlier, and support candidate selection during discovery and preclinical development.

 

Metabolism & Stability Assessment

In vitro assays supporting evaluation of metabolic stability, intrinsic clearance, and compound behavior across biological systems.

  • Liver microsome stability assays
  • Hepatocyte stability studies
  • Plasma stability evaluation
  • Intrinsic clearance assessment

Drug Interaction Evaluation

Capabilities supporting assessment of drug-drug interaction risk and transporter-related liabilities during discovery.

  • CYP450 inhibition studies
  • CYP induction assays
  • Transporter interaction studies

Discovery-Focused Decision Support

ADME data helping teams prioritize compounds, improve exposure profiles, and guide medicinal chemistry optimization.

  • Early liability identification
  • Structure–property relationship support
  • Candidate selection guidance

Metabolic Stability Studies

Microsomal, hepatocyte, and plasma stability studies.

CYP450 Inhibition & Induction

Assessment of cytochrome P450 interaction potential.

Plasma Protein Binding

Evaluation of compound binding and free fraction.

Transporter Interaction Studies

Assessment of uptake and efflux transporter interactions.

Download the In Vitro ADME Overview

Explore BioDuro’s in vitro ADME capabilities supporting metabolism, stability, transporter interaction, and pharmacokinetic evaluation across discovery programs.